Synthesis of novel N- and C-acyclic nucleosides derived from 2-hydrazino-6-methyluracil
نویسندگان
چکیده
منابع مشابه
synthesis of sulfides from alcohols and thiols in solvent-freeconditions and deoxygenation of sulfoxides
کاتالیست یک سنتز جدید برای تیواترها توصیف شده است. واکنش الکل ها با آریل، هتروآریل و آلکیل تیو ل ها درحضور 1،3،5- تری آزو- 2،4،6- تری فسفرین-2،2،4،4،6،6 هگزاکلراید ((tapc به عنوان یک کاتالیست موُثر، بازده های خوب تا عالی از تیواترها را حاصل می کند. علاوه براین، واکنش تحت شرایط بدون فلز و بدون حلال پیش می رود، بنابراین یک مکمل جالب برای روش های شناخته شده سنتز تیواترها ارائه می دهد. یک مکانیسم ا...
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A series of novel 2-substituted hydrazino-6-fluoro-1,3-benzothiazole derivatives were synthesized by synthesizing the 2-hydrazino-6-fluorobenzothiazole and refluxing of this with different substituted acetophenones. The synthesized compounds were evaluated for their possible antimicrobial activity. The structures of few representative compounds were elucidated by IR and NMR. For present work ef...
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Carbocyclic nucleoside analogues remain interesting target molecules having the potential to combine biological activity with greater metabolic stability than their sugar counterparts. This paper describes a rapid and versatile synthetic approach to such compounds based on commercial cyclopentenones (e.g., 1) that has been developed in our laboratory. Carbocyclic nucleosides like 2 0-methylaris...
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ژورنال
عنوان ژورنال: Egyptian Journal of Chemistry
سال: 2020
ISSN: 2357-0245
DOI: 10.21608/ejchem.2020.21459.2279